, Chem. Res.Toxicol. Chem. Res. Toxicol, vol.2012, issue.25, pp.532-542, 2012.
, Angew. Chem. Int. Ed. Angew. Chem. Int. Ed. Chem. Rev. Nature, vol.57, issue.529, pp.1758-1784, 2008.
DOI: 10.1126/science, Angew. Chem. Int. Ed, vol.534, pp.230-234, 2014. ,
C???H Functionalisation for Hydrogen Isotope Exchange, Angewandte Chemie International Edition, vol.529, issue.12, pp.3022-3047, 2018. ,
DOI : 10.1038/nature16464
Preparation of Compounds Labeled with Tritium and Carbon-14, Process Res. Dev. 2014, pp.4545-4553, 2009. ,
C-11 Radiochemistry in Cancer Imaging Applications, Current Topics in Medicinal Chemistry, vol.10, issue.11, pp.1060-1095, 2010. ,
DOI : 10.2174/156802610791384261
C???O bonds made easily for positron emission tomography radiopharmaceuticals, Chemical Society Reviews, vol.18, issue.17, pp.4708-4726, 2016. ,
DOI : 10.1002/chem.201103128
, For recent labeling methods using [ 11 C]CN -, see: a) K, J. Makaravage
, Chem. Commun, vol.20, issue.53, pp.1530-1533, 2017.
, J. Am. Chem. Soc, vol.137, pp.648-651, 2015.
, For recent labeling methods using [ 11 C]CO2, see: a)
, Angew. Chem. Int. Ed, vol.48, pp.3482-3485, 2009.
, Angew. Chem. Int. Ed, vol.2012, issue.51, pp.2698-2702
, Bioconjugate Chem, vol.27, pp.1382-1389, 2016.
The therapeutic journey of benzimidazoles: A review, Bioorganic & Medicinal Chemistry, vol.20, issue.21, pp.6208-6236, 2000. ,
DOI : 10.1016/j.bmc.2012.09.013
, Angew. Chem. Int. Ed, vol.54, pp.10313-10316, 2015.
Synthesis of 1-(2-ethoxyethyl)-2-(4-methyl-1-homopiperazinyl)-[2-14C]benzimidazole difumarate([14C]KB-2413), Journal of Labelled Compounds and Radiopharmaceuticals, vol.34, issue.II, pp.331-338, 1987. ,
DOI : 10.1002/jlcr.2580240314
C-radiolabelled ureas, Journal of Labelled Compounds and Radiopharmaceuticals, vol.26, issue.4, pp.202-208, 2014. ,
DOI : 10.1002/zfch.19860261214
, It is worth noting that no examples of cyclic ureas were reported with this method, Chem. Eur. J, vol.17, pp.259-264, 2011.
, Acc. Chem. Res. Angew. Chem. Int. Ed, vol.44, issue.50, pp.666-676, 2011.
This report describe that [ 11 C]phenylisocyanate could be produced by trapping [ 11 C]CO2 in a solution of phenyltriphenylphosphinimine. The method was applied on four linear substrates with moderate yelds and may be constrained by the lack of structurally diverse triphenylphosphinimines, Tang, N. Jiao, J. Am. Chem. Soc. Chem. Commun. J. Org. Chem, vol.49, issue.82, pp.321-330, 2006. ,
, Oxatomide was previously labeled at the same position using [ 14 C]-urea in much more drastic conditions, Interestingly °C
Plasma levels, biotransformation and excretion of oxatomide (R 35 443) in rats, dogs and man, Xenobiotica, vol.18, issue.6, pp.445-362, 1984. ,
DOI : 10.1007/BF03189515
F]-PET Imaging in a Primate Brain, Journal of Medicinal Chemistry, vol.58, issue.20, pp.8066-8096, 2015. ,
DOI : 10.1021/acs.jmedchem.5b00874
URL : https://hal.archives-ouvertes.fr/hal-02068052
Preparation and pharmaceutical evaluation for clinical application of high specific activity S-(???)[11C]CGP-12177, a radioligand for ??-adrenoreceptors, Nuclear Medicine Communications, vol.25, issue.8, pp.845-849, 2004. ,
DOI : 10.1097/01.mnm.0000134320.39903.75
, J. Am. Chem. Soc. Angew. Chem. Int. Ed, vol.17, issue.56, pp.354-357, 2015.